Acetaminophen Tolperisone
Acetaminophen/Tolperisone is a combination medication that pairs an analgesic with a muscle relaxant to address both pain and associated muscle tension. This multi-ingredient formulation is typically used for musculoskeletal conditions involving both discomfort and involuntary muscle contractions. The combination aims to provide more comprehensive symptom relief than either component alone.
A combination analgesic and muscle relaxant used for pain with muscle spasms.
Key facts at a glance
- RxNorm
- 1007030
- Generic
- Acetaminophen / Tolperisone
- Class
- multi-ingredient
- Brands
- —
- Availability
- rx
- Lactation
- unknown
- Routes
- —
- Forms
- —
- Regions
- US, EU, CN, JP
- Monitoring
- —
This page is for informational purposes only.
Do not use this information to diagnose yourself or to replace a physician's advice. Always consult a qualified healthcare provider before starting, stopping, or changing any medication. If you believe you are experiencing a medical emergency, call your local emergency number immediately.
Used for musculoskeletal pain conditions involving muscle spasms, such as back pain, neck pain, and other acute or chronic painful musculoskeletal disorders with associated muscle tension.
Acetaminophen provides pain relief and fever reduction through central prostaglandin inhibition, while tolperisone acts on the central nervous system to reduce muscle hyperactivity and spasms by modulating nerve transmission in spinal cord and brainstem pathways.
Should be used with caution in patients with liver disease due to the acetaminophen component; alcohol should be avoided during treatment. Tolperisone may cause drowsiness or dizziness in some patients. As with all combination medications, patients should be aware of potential side effects from both components and use only as directed by a healthcare provider.
Official drug label
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This information is for educational purposes only and is not a substitute for professional medical advice, diagnosis, or treatment.
This content is for general informational and educational purposes only and is not a substitute for professional medical advice, diagnosis, or treatment. Always seek the guidance of a qualified healthcare provider with any questions you have about a medical condition, and never disregard professional medical advice or delay seeking it because of something you read here.
If you think you may have a medical emergency, call your local emergency number or go to the nearest emergency department immediately.
Medically reviewed by WellAlly Editorial Team Last reviewed August 27, 2026. · Read our editorial policy