Nebivolol
Bystolic (nebivolol) is a prescription beta-blocker used to treat high blood pressure. It works by blocking the effects of adrenaline on the heart, allowing it to beat more slowly and with less force, while also promoting blood vessel relaxation. This medication is typically prescribed for adults with hypertension to help reduce the risk of heart attacks and strokes.
Bystolic is a beta-blocker medication used to treat high blood pressure by reducing heart rate and relaxing blood vessels.
Key facts at a glance
- RxNorm
- 751613
- Generic
- Bystolic
- Class
- brand-name
- Brands
- —
- Availability
- rx
- Lactation
- unknown
- Routes
- —
- Forms
- —
- Regions
- US, EU, CN, JP
- Monitoring
- —
This page is for informational purposes only.
Do not use this information to diagnose yourself or to replace a physician's advice. Always consult a qualified healthcare provider before starting, stopping, or changing any medication. If you believe you are experiencing a medical emergency, call your local emergency number immediately.
Bystolic is FDA-approved for the treatment of hypertension (high blood pressure) in adults. It may be used alone or in combination with other blood pressure medications. Managing high blood pressure helps reduce the risk of serious cardiovascular events such as heart attack and stroke.
Bystolic is a beta-1 selective adrenergic receptor blocker, meaning it primarily targets receptors in the heart to reduce heart rate and the force of contractions. Additionally, it stimulates the release of nitric oxide from blood vessel linings, causing vasodilation (widening of blood vessels), which further helps lower blood pressure.
Bystolic should not be stopped abruptly, as sudden discontinuation may worsen chest pain or trigger a heart attack. Common side effects may include headache, fatigue, and dizziness. Patients with certain heart conditions, liver impairment, or who are taking other blood pressure medications should discuss their full medical history with their healthcare provider before starting Bystolic.
Official drug label
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This information is for educational purposes only and is not a substitute for professional medical advice, diagnosis, or treatment.
This content is for general informational and educational purposes only and is not a substitute for professional medical advice, diagnosis, or treatment. Always seek the guidance of a qualified healthcare provider with any questions you have about a medical condition, and never disregard professional medical advice or delay seeking it because of something you read here.
If you think you may have a medical emergency, call your local emergency number or go to the nearest emergency department immediately.
Medically reviewed by WellAlly Editorial Team Last reviewed September 3, 2026. · Read our editorial policy