Ceftaroline Fosamil Acetate
Ceftaroline Fosamil Acetate is a fifth-generation cephalosporin antibiotic that works by inhibiting bacterial cell wall synthesis. It is used to treat acute bacterial skin and skin structure infections (ABSSSI) and community-acquired bacterial pneumonia (CABP) in adults. This medication has activity against certain gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA).
Ceftaroline Fosamil Acetate is a cephalosporin antibiotic used to treat certain serious skin infections and pneumonia caused by susceptible bacteria.
Key facts at a glance
- RxNorm
- 1743286
- Generic
- Ceftaroline Fosamil Acetate
- Class
- pin-variant
- Brands
- —
- Availability
- rx
- Lactation
- unknown
- Routes
- —
- Forms
- —
- Regions
- US, EU, CN, JP
- Monitoring
- —
This page is for informational purposes only.
Do not use this information to diagnose yourself or to replace a physician's advice. Always consult a qualified healthcare provider before starting, stopping, or changing any medication. If you believe you are experiencing a medical emergency, call your local emergency number immediately.
Treats acute bacterial skin and skin structure infections (ABSSSI) and community-acquired bacterial pneumonia (CABP) caused by susceptible gram-positive and gram-negative bacteria. Particularly notable for activity against MRSA and other resistant organisms.
Binds to penicillin-binding proteins (PBPs), particularly PBP2a in resistant organisms, inhibiting transpeptidation during cell wall synthesis. This weakens the bacterial cell wall, leading to cell death.
Administered intravenously. Should be used only for confirmed or suspected bacterial infections. May cause hypersensitivity reactions, including anaphylaxis. Common side effects include nausea, rash, and diarrhea. Patients with known cephalosporin or penicillin allergies should use with caution. Safety in pregnancy and breastfeeding should be discussed with a healthcare provider.
Official drug label
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This information is for educational purposes only and is not a substitute for professional medical advice, diagnosis, or treatment.
This content is for general informational and educational purposes only and is not a substitute for professional medical advice, diagnosis, or treatment. Always seek the guidance of a qualified healthcare provider with any questions you have about a medical condition, and never disregard professional medical advice or delay seeking it because of something you read here.
If you think you may have a medical emergency, call your local emergency number or go to the nearest emergency department immediately.
Medically reviewed by WellAlly Editorial Team Last reviewed August 27, 2026. · Read our editorial policy