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Cerivastatin Sodium

Published: July 26, 2026Updated: August 25, 2026

Cerivastatin Sodium was a cholesterol-lowering medication belonging to the statin drug class. It worked by inhibiting HMG-CoA reductase, an enzyme involved in cholesterol synthesis in the liver. This medication was prescribed to patients with hyperlipidemia to reduce elevated cholesterol and triglyceride levels.

Quick summary

Cerivastatin was a statin medication for high cholesterol that was withdrawn from the market in 2001 due to safety concerns.

Medically reviewed by WellAlly Editorial TeamLast reviewed August 25, 2026Editorial policy

Key facts at a glance

RxNorm
221072
Generic
Cerivastatin Sodium
Class
pin-variant
Brands
—
Availability
rx
Lactation
unknown
Routes
—
Forms
—
Regions
US, EU, CN, JP
Monitoring
—

This page is for informational purposes only.

Do not use this information to diagnose yourself or to replace a physician's advice. Always consult a qualified healthcare provider before starting, stopping, or changing any medication. If you believe you are experiencing a medical emergency, call your local emergency number immediately.

Treatment of hypercholesterolemia and mixed dyslipidemia to lower total cholesterol, LDL cholesterol, and triglyceride levels. Was used when diet and exercise modifications were insufficient.

Cerivastatin is an HMG-CoA reductase inhibitor (statin) that blocks the enzyme responsible for cholesterol synthesis in the liver, reducing overall cholesterol production and increasing LDL receptor activity.

Cerivastatin was voluntarily withdrawn from the market worldwide in August 2001 due to unacceptable risk of serious rhabdomyolysis (muscle breakdown), particularly when used in combination with gemfibrozil. This resulted in multiple deaths. The medication is no longer available for prescription use. Patients were advised to consult their healthcare providers for alternative cholesterol management options.

Official drug label

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This information is for educational purposes only and is not a substitute for professional medical advice, diagnosis, or treatment.

Medical Disclaimer

This content is for general informational and educational purposes only and is not a substitute for professional medical advice, diagnosis, or treatment. Always seek the guidance of a qualified healthcare provider with any questions you have about a medical condition, and never disregard professional medical advice or delay seeking it because of something you read here.

If you think you may have a medical emergency, call your local emergency number or go to the nearest emergency department immediately.

Medically reviewed by WellAlly Editorial Team Last reviewed August 25, 2026. · Read our editorial policy