Pentobarbital, Carbromal
Pentobarsol is a brand-name barbiturate medication used primarily for sedation, anesthesia induction, and seizure management in clinical settings. It works by enhancing the effects of GABA in the central nervous system, resulting in decreased neuronal activity. This medication requires close medical supervision due to its narrow therapeutic index and potential for dependence.
Pentobarsol is a barbiturate used for sedation and anesthesia that acts on GABA receptors in the brain.
Key facts at a glance
- RxNorm
- 2626488
- Generic
- Pentobarsol
- Class
- brand-name
- Brands
- —
- Availability
- rx
- Lactation
- unknown
- Routes
- —
- Forms
- —
- Regions
- US, EU, CN, JP
- Monitoring
- —
This page is for informational purposes only.
Do not use this information to diagnose yourself or to replace a physician's advice. Always consult a qualified healthcare provider before starting, stopping, or changing any medication. If you believe you are experiencing a medical emergency, call your local emergency number immediately.
Pentobarsol is used for procedural sedation, induction of anesthesia, and control of certain seizure disorders in healthcare settings.
As a barbiturate, Pentobarsol enhances the effect of gamma-aminobutyric acid (GABA) at GABA-A receptors, leading to increased inhibitory signaling and decreased neuronal excitability in the central nervous system.
Pentobarsol is a Schedule II controlled substance with a narrow therapeutic window. It requires administration by qualified healthcare professionals with resuscitation equipment available. Risks include respiratory depression, dependence, and potentially fatal overdose when combined with other CNS depressants. Close hemodynamic monitoring is essential during use.
Official drug label
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This information is for educational purposes only and is not a substitute for professional medical advice, diagnosis, or treatment.
This content is for general informational and educational purposes only and is not a substitute for professional medical advice, diagnosis, or treatment. Always seek the guidance of a qualified healthcare provider with any questions you have about a medical condition, and never disregard professional medical advice or delay seeking it because of something you read here.
If you think you may have a medical emergency, call your local emergency number or go to the nearest emergency department immediately.
Medically reviewed by WellAlly Editorial Team Last reviewed July 26, 2026. · Read our editorial policy